انواع ضدآندروژن و مقدار مصرف:
|
,1 mg(0.2 ml) a day S.C |
Lupron (Tap pharmaceyticals Usa: 14 mg/2.8 ml vials) |
Leuprolide acetate |
|
0.5 mg every 8h, S.C. tor 7 days, then bilateral nasal spray beto before and after the 3 meals a day (= 12 inhalations) |
Super fact, Inject able and nasal (Hoechst) |
Buserelin |
|
1000 mg 2/week i.m. |
USA: Delautin |
Hydroxyprogestrone capraote |
|
100-200 orally on alternate days 500mg/day i.m. 200-300 mg/day orally (Endometrial canser) |
USA: Provera, Depo. Provera |
Medroxyprogestrone acetate |
|
160 mg/day in 4 divided doses 40-320 mg/day orally in divided doses |
Megace ( mead Johnson, USA: 20 and 40 mg tablets) |
Megestrol acetate |
|
10-20 mg orally twice daily |
USA: Nolvadex, Stuart Pharmaceutical |
Tamoxifen |
|
250 mg x 2-4/day Administer adrenal replacement therapy (hydrocortisone: 40-50 mg/day in divided doses) |
USA: Cytraden,Ciba Geigy |
Aminoglutethimide |
عوارض : تهوع، خونريزي رحمي ، اختلال قاعدگي ، درد استخوان در محل تومور ، رتينوپاتي ، سرگيجه ، ادم ، کلستاز ، سرکوب مغز استخوان